Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
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Sigma non-opioid intracellular receptor 1 (Homo sapiens (Human)) | BDBM50022721 ((R)-amphetamine | AMPHETAMINE | CHEMBL19393) | PDB UniProtKB/SwissProt antibodypedia GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 4.64E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Virginia Commonwealth University Curated by ChEMBL | Assay Description Binding affinity towards sigma opioid receptor in guinea pig cerebral homogenate using [3H]DTG as radioligand | J Med Chem 34: 1094-8 (1991) BindingDB Entry DOI: 10.7270/Q28C9WV8 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] B (Rattus norvegicus (rat)) | BDBM50022721 ((R)-amphetamine | AMPHETAMINE | CHEMBL19393) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.80E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Syntex Research Curated by ChEMBL | Assay Description Competitive inhibition of Rat liver Monoamine Oxidase B at 37 degree C (pH= 7.4) | J Med Chem 31: 1558-66 (1988) BindingDB Entry DOI: 10.7270/Q21J9BCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] B (Bos taurus) | BDBM50022721 ((R)-amphetamine | AMPHETAMINE | CHEMBL19393) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 3.80E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Syntex Research Curated by ChEMBL | Assay Description Inhibitory activity against Monoamine Oxidase B of Bovine liver in competitive inhibition assay at 25 degree C (pH=7.4) | J Med Chem 31: 1558-66 (1988) BindingDB Entry DOI: 10.7270/Q21J9BCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Amine oxidase [flavin-containing] B (Rattus norvegicus (rat)) | BDBM50022721 ((R)-amphetamine | AMPHETAMINE | CHEMBL19393) | PDB MMDB KEGG UniProtKB/SwissProt B.MOAD GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 7.60E+5 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Syntex Research Curated by ChEMBL | Assay Description In vitro inhibition of bovine monoamine oxidase B. | J Med Chem 31: 1558-66 (1988) BindingDB Entry DOI: 10.7270/Q21J9BCX | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phenylethanolamine N-methyltransferase (Bos taurus (bovine)) | BDBM50022721 ((R)-amphetamine | AMPHETAMINE | CHEMBL19393) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.38E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
University of Kansas Curated by ChEMBL | Assay Description In vitro binding affinity of compound towards bovine adrenal phenylethanolamine N-methyl-transferase (PNMT) | J Med Chem 31: 1984-6 (1988) BindingDB Entry DOI: 10.7270/Q2QF8TFD | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Phenylethanolamine N-methyltransferase (Bos taurus (bovine)) | BDBM50022721 ((R)-amphetamine | AMPHETAMINE | CHEMBL19393) | PDB UniProtKB/SwissProt GoogleScholar AffyNet | Purchase CHEMBL KEGG PC cid PC sid PDB UniChem Patents Similars | PubMed | 1.38E+6 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
TBA Curated by ChEMBL | Assay Description Inhibitory activity against bovine adrenal norepinephrine N-methyl-transferase was determined | J Med Chem 25: 1248-50 (1983) BindingDB Entry DOI: 10.7270/Q2S46SJ3 | |||||||||||
More data for this Ligand-Target Pair |